Author

Shoji Fukumoto

Observed names: Fukumoto, Shoji, Shoji FUKUMOTO

Institutions: Japan Tobacco (Japan), Takeda (Japan)

Observed institutions: Japan Tobacco (Japan), Takeda (Japan), Kobe University

OpenAlex ID: A5113568290

Identification of Benzoxazin-3-one Derivatives as Novel, Potent, and Selective Nonsteroidal Mineralocorticoid Receptor Antagonists

2011 · Tomoaki Hasui, Nobuyuki Matsunaga, et al. · Journal of Medicinal Chemistry · 117

Discovery, synthesis and biological evaluation of isoquinolones as novel and highly selective JNK inhibitors (2)

2008 · Yasutomi Asano, Shuji Kitamura, et al. · Bioorganic & Medicinal Chemistry · 93

Design, Synthesis, and Evaluation of the Highly Selective and Potent G-Protein-Coupled Receptor Kinase 2 (GRK2) Inhibitor for the Potential Treatment of Heart Failure

2017 · Tomohiro Okawa, Yoshio Aramaki, et al. · Journal of Medicinal Chemistry · 62

Novel, Non-acylguanidine-type Na+/H+ Exchanger Inhibitors: Synthesis and Pharmacology of 5-Tetrahydroquinolinylidene Aminoguanidine Derivatives

2002 · Shoji Fukumoto, Eiko Imamiya, et al. · Journal of Medicinal Chemistry · 51

Discovery of an Orally Bioavailable, Brain-Penetrating, in Vivo Active Phosphodiesterase 2A Inhibitor Lead Series for the Treatment of Cognitive Disorders

2017 · Satoshi Mikami, Shigekazu Sasaki, et al. · Journal of Medicinal Chemistry · 45

Design, synthesis, and structure–activity relationships of dihydrofuran-2-one and dihydropyrrol-2-one derivatives as novel benzoxazin-3-one-based mineralocorticoid receptor antagonists

2013 · Tomoaki Hasui, Taiichi Ohra, et al. · Bioorganic & Medicinal Chemistry · 36

Discovery of 6-[5-(4-fluorophenyl)-3-methyl-pyrazol-4-yl]-benzoxazin-3-one derivatives as novel selective nonsteroidal mineralocorticoid receptor antagonists

2014 · Tomoaki Hasui, Norio Ohyabu, et al. · Bioorganic & Medicinal Chemistry · 30

In vitro and in vivo pharmacology of a structurally novel Na+‐H+ exchange inhibitor, T‐162559

2002 · Keiji Kusumoto, Hideki Igata, et al. · British Journal of Pharmacology · 26

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Potent and selective inhibition of the human Na+/H+ exchanger isoform NHE1 by a novel aminoguanidine derivative T-162559

2001 · Tomohiro Kawamoto, Hiroyuki Kimura, et al. · European Journal of Pharmacology · 22

Discovery of orally efficacious RORγt inverse agonists. Part 2: Design, synthesis, and biological evaluation of novel tetrahydroisoquinoline derivatives

2017 · Mitsunori Kono, Tsuneo Oda, et al. · Bioorganic & Medicinal Chemistry · 21

Titanium Trichloride Mediated Reduction of Nitrostyrenes

1986 · Akira Sera, Shoji Fukumoto, et al. · Heterocycles · 18

Titanium(III) Chloride Mediated Reduction of 1-Nitro-2-phenylethenes

1991 · Akira Sera, Shoji Fukumoto, et al. · Bulletin of the Chemical Society of Japan · 15

Synthesis and thromboxane A2/prostaglandin H2 receptor antagonistic activity of phenol derivatives

1992 · Shoji Fukumoto, Mitsuru Shiraishi, et al. · Journal of Medicinal Chemistry · 12

Direct and enantiospecific ortho-benzylation of phenols by the Mitsunobu reaction

1996 · Shoji Fukumoto, Shigeha Fukushi, et al. · Journal of the Chemical Society Perkin Transactions 1 · 10

Design and Synthesis of Conformationally Constrained RORγt Inverse Agonists

2019 · Ayumu Sato, Yoshiyuki Fukase, et al. · ChemMedChem · 8

Practical application of 3-substituted-2,6-difluoropyridines in drug discovery: Facile synthesis of novel protein kinase C theta inhibitors

2017 · Taisuke Katoh, Yoshihide Tomata, et al. · Bioorganic & Medicinal Chemistry Letters · 8

Stereoselective Synthesis and Thromboxane A2 (TXA2) Receptor Antagonistic Activity of Optically Active Phenol Derivatives.

1996 · Shoji FUKUMOTO, Zen-ichi TERASHITA, et al. · Chemical and Pharmaceutical Bulletin · 4

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CCDC 1575732: Experimental Crystal Structure Determination

2017 · Kono, Mitsunori, Oda, Tsuneo, et al. · The Cambridge Structural Database

In vitro and in vivo pharmacology of a non-acylguanidine Na-H exchange inhibitor,T 162559

2001 · Keiji Kusumoto, Hideki Igata, et al. · Journal of Molecular and Cellular Cardiology

Synthesis and Txa_2/pgh_2 Receptor Antagonistic Activity of Phenol Derivatives

1991 · Shoji Fukumoto, Mitsuru Shiraishi, et al. · Journal of Pharmacobio-Dynamics

Works count: 20

Citation count: 578

H-index: 12

I10-index: 14