Discovery of 6-[5-(4-fluorophenyl)-3-methyl-pyrazol-4-yl]-benzoxazin-3-one derivatives as novel selective nonsteroidal mineralocorticoid receptor antagonists
Year: 2014
Type: article
Source: Bioorganic & Medicinal Chemistry
Authors: Tomoaki Hasui, Norio Ohyabu, Taiichi Ohra, Koji Fuji, Takahiro Sugimoto, Jun Fujimoto, Kouhei Asano, Masato Oosawa, Sachiko Shiotani, Nobuhiro Nishigaki, Keiji Kusumoto, Hideki Matsui, Atsushi Mizukami, Noriyuki Habuka, Satoshi Sogabe, Satoshi Endo, Midori Ono, Christopher S. Siedem, Tony P. Tang, Cassandra Gauthier, Lisa A. De Meese, Steven A. Boyd, Shoji Fukumoto
Institutions: Takeda (Japan), Array BioPharma (United States)
Language: English
Subfield: Endocrinology, Diabetes and Metabolism
Field: Medicine
Domain: Health Sciences
Open Access status: closed
OpenAlex ID: W2018942927
