Get started
Author

Akito Yasuhara

Observed name: Akito YASUHARA
OpenAlex ID: A5113821169
MGS0039: a potent and selective group II metabotropic glutamate receptor antagonist with antidepressant-like activity
2003 · Shigeyuki Chaki, Ryoko Yoshikawa, et al. · Neuropharmacology · 262
Novel synthetic strategy of carbolines via palladium-catalyzed amination and arylation reaction
1999 · Takehiko Iwaki, Akito Yasuhara, et al. · Journal of the Chemical Society Perkin Transactions 1 · 158
Convenient synthesis of 2-substituted indoles from 2-ethynylanilines with tetrabutylammonium fluoride
1999 · Akito Yasuhara, Yuichi Kanamori, et al. · Journal of the Chemical Society Perkin Transactions 1 · 109
Deprotection of N-sulfonyl nitrogen-heteroaromatics with tetrabutylammonium fluoride
1998 · Akito Yasuhara, Takao Sakamoto · Tetrahedron Letters · 101
Cyclization reactions of 2-alkynylbenzyl alcohol and 2-alkynylbenzylamine derivatives promoted by tetrabutylammonium fluoride
2001 · Kou Hiroya, Rumi Jouka, et al. · Tetrahedron · 90
Total syntheses of three natural products, vignafuran, 2-(4-hydroxy-2-methoxyphenyl)-6-methoxybenzofuran-3-carboxylic acid methyl ester, and coumestrol from a common starting material
2000 · Kou Hiroya, Naoyuki Suzuki, et al. · Journal of the Chemical Society Perkin Transactions 1 · 86
Selective Monodesulfonylation of N,N-Disulfonylarylamines with Tetrabutylammonium Fluoride.
1999 · Akito YASUHARA, Mitsuyoshi KAMEDA, et al. · Chemical and Pharmaceutical Bulletin · 81
PDF
Neuropharmacological profiles of antagonists of group II metabotropic glutamate receptors
2005 · Naoya Kawashima, Jun-ichi Karasawa, et al. · Neuroscience Letters · 66
Preparation of Ethyl Arylpropiolates from Aryl Iodides by Palladium-Catalyzed Cross-Coupling Reaction
1992 · Takao Sakamoto, Futoshi Shiga, et al. · Synthesis · 61
Synthesis, in Vitro Pharmacology, Structure−Activity Relationships, and Pharmacokinetics of 3-Alkoxy-2-amino-6-fluorobicyclo[3.1.0]hexane-2,6-dicarboxylic Acid Derivatives as Potent and Selective Group II Metabotropic Glutamate Receptor Antagonists
2004 · Atsuro Nakazato, Kazunari Sakagami, et al. · Journal of Medicinal Chemistry · 60
Synthesis of 2,3-Disubstituted Indole Using Palladium(II)-Catalyzed Cyclization with Alkenylation Reaction.
2002 · Akito Yasuhara, Yousuke Takeda, et al. · Chemical and Pharmaceutical Bulletin · 57
PDF
Synthesis of 2-Substituted 3-Alkenyl-indoles by the Palladium-catalyzed Cyclization Followed by Alkenylation (Heck Reaction)
1998 · Takao Sakamoto, Akito Yasuhara, et al. · Heterocycles · 56
Condensed heteroaromatic ring systems. XVIII. Palladium-catalyzed cross-coupling reaction of aryl bromides with (Z)-1-ethoxy-2-tributylstannylethene and its utilization for construction of condensed heteroaromatics
1991 · Takao Sakamoto, Yoshinori Kondo, et al. · Tetrahedron · 52
Convenient Indole Synthesis from 2-Iodoanilines and Terminal Alkynes by the Sequential Sonogashira Reaction and the Cyclization Reaction Promoted by Tetrabutylammonium Fluoride (TBAF)
2003 · Naoyuki Suzuki, Sakura Yasaki, et al. · Chemical and Pharmaceutical Bulletin · 45
PDF
An Efficient Method for the Deallylation of Allyl Aryl Ethers Using Electrochemically Generated Nickel
1999 · Akito Yasuhara, Atsushi Kasano, et al. · The Journal of Organic Chemistry · 44
Prodrugs of 3-(3,4-dichlorobenzyloxy)-2-amino-6-fluorobicyclo[3.1.0]hexane-2,6-dicarboxylic acid (MGS0039): A potent and orally active group II mGluR antagonist with antidepressant-like potential
2006 · Akito Yasuhara, Masato Nakamura, et al. · Bioorganic & Medicinal Chemistry · 43
Convenient Reduction of Nitrobenzenes to Anilines Using Electrochemically Generated Nickel
1999 · Akito Yasuhara, Atsushi Kasano, et al. · The Journal of Organic Chemistry · 41
Neurophysiologic and Antipsychotic Profiles of TASP0433864, a Novel Positive Allosteric Modulator of Metabotropic Glutamate 2 Receptor
2014 · Tetsuaki Hiyoshi, Toshiyuki Marumo, et al. · Journal of Pharmacology and Experimental Therapeutics · 34
A Concise Synthesis of Furostifoline by Tetrabutylammonium Fluoride-Promoted Indole Ring Formation.
2002 · Akito Yasuhara, Naoyuki Suzuki, et al. · Chemical and Pharmaceutical Bulletin · 34
PDF
Condensed Heteroaromatic Ring Systems. XXIII. A Concise Synthesis of Hippadine
1993 · Takao Sakamoto, Akito Yasuhara, et al. · Heterocycles · 34
Metabotropic Glutamate Receptors: Potential Drug Targets for Psychiatric Disorders
2010 · Akito Yasuhara, Shigeyuki Chaki · The Open Medicinal Chemistry Journal · 33
PDF
Synthesis of Ethoxyethynylarenes by the Palladium-Catalyzed Reaction of Aryl Iodides with Ethoxy(trialkylstannyl)acetylenes.
1994 · Takao SAKAMOTO, Akito YASUHARA, et al. · Chemical and Pharmaceutical Bulletin · 29
PDF
Convenient indole synthesis from ethynylanilines with a polymer-supported fluoride
2002 · Akito Yasuhara, Naoyuki Suzuki, et al. · Tetrahedron Letters · 26
Palladium-Catalyzed Cross-Coupling Reaction of Ethoxy(tributylstannyl)acetylene with Aryl Iodides
1992 · Takao Sakamoto, Akito Yasuhara, et al. · Synlett · 25
Antipsychotic profiles of TASP0443294, a novel and orally active positive allosteric modulator of metabotropic glutamate 2 receptor
2015 · Hirohiko Hikichi, Tetsuaki Hiyoshi, et al. · Journal of Pharmacological Sciences · 24
PDF
Works count: 45
Citation count: 1,738
H-index: 24
I10-index: 29
Year
Topic
Type