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Discovery of inhibitors of the mitotic kinase TTK based on N-(3-(3-sulfamoylphenyl)-1H-indazol-5-yl)-acetamides and carboxamides

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Year: 2014
Type: article
Source: Bioorganic & Medicinal Chemistry
DOI: 10.1016/j.bmc.2014.06.027
Authors: Radoslaw Laufer, Grace Ng, Yong Liu, Narendra Kumar B. Patel, Louise G. Edwards, Yunhui Lang, Sze-Wan Li, Miklos Feher, Don E. Awrey, Genie Leung, Irina Beletskaya, Olga Plotnikova, Jacqueline M. Mason, Richard Hodgson, Xin Wei, Guodong Mao, Xunyi Luo, Ping Huang, Erin Green, Reza Kiarash, Dan Chi-Chia Lin, Marees Harris-Brandts, Fuqiang Ban, Vincent Nadeem, Tak W. Mak, Guohua J. Pan, Wei Qiu, Nickolay Y. Chirgadze, Henry W. Pauls
Institutions: University Health Network, Campbell Family Institute for Breast Cancer Research, Princess Margaret Cancer Centre
Language: English

Topic: Heterocyclic Compound Synthesis and Bioactivity
Subfield: Organic Chemistry
Field: Chemistry
Domain: Physical Sciences
SDG: Good health and well-being

Open Access status: closed

Funders: Shionogi, Argonne National Laboratory
OpenAlex ID: W1990899207
FWCI: 2.714
Cites: 50
Cited by: 42
Related to: 10
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