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Discovery of CS-2100, a potent, orally active and S1P3-sparing S1P1 agonist

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Year: 2012
Type: article
Source: Bioorganic & Medicinal Chemistry Letters
DOI: 10.1016/j.bmcl.2011.12.019
Authors: Tsuyoshi Nakamura, Masayoshi Asano, Yukiko Sekiguchi, Yumiko Mizuno, Kazuhiko Tamaki, Takako Kimura, Futoshi Nara, Yumi Kawase, Takaichi Shimozato, Hiromi Doi, Takashi Kagari, Wataru Tomisato, Ryotaku Inoue, Miyuki Nagasaki, Hiroshi Yuita, Keiko Oguchi-Oshima, Reina Kaneko, Nobuaki Watanabe, Yasuyuki Abe, Takahide Nishi
Institution: Daiichi-Sankyo (Japan)
Language: English

Topic: Sphingolipid Metabolism and Signaling
Subfield: Molecular Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: closed
OpenAlex ID: W2020199692
FWCI: 1.434
Cites: 28
Cited by: 24
Related to: 10
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