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Discovery of a First-in-Class Receptor Interacting Protein 1 (RIP1) Kinase Specific Clinical Candidate (GSK2982772) for the Treatment of Inflammatory Diseases

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Year: 2017
Type: other
Source: Journal of Medicinal Chemistry
DOI: 10.1021/acs.jmedchem.6b01751
Authors: Philip A. Harris, Scott B. Berger, Jae U. Jeong, Rakesh Nagilla, Deepak Bandyopadhyay, Nino Campobasso, Carol A. Capriotti, Julie A. Cox, Lauren Dare, Xiaoyang Dong, Patrick M. Eidam, Joshua N. Finger, Sandra J. Hoffman, James Kang, Viera Kasparcova, Bryan W. King, Ruth Lehr, Yunfeng Lan, Lara K. Leister, John D. Lich, Thomas T. MacDonald, Nathan A. Miller, Michael T. Ouellette, Christina S. Pao, Attiq Rahman, Michael A. Reilly, Alan R. Rendina, Elizabeth J. Rivera, Michelle C. Schaeffer, Clark A. Sehon, Robert R. Singhaus, Helen H. Sun, Barbara A. Swift, Rachel D. Totoritis, Anna Vossenkämper, Paris Ward, David D. Wisnoski, Daohua Zhang, Robert W. Marquis, Peter J. Gough, John Bertin
Institutions: GlaxoSmithKline (United States), Queen Mary University of London, Blizard Institute
Language: English

Topic: Cell death mechanisms and regulation
Subfield: Molecular Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: closed
OpenAlex ID: W2584580415
Cites: 30
Cited by: 509
Related to: 10
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