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Pyrrolobenzodiazepine Dimer Antibody–Drug Conjugates: Synthesis and Evaluation of Noncleavable Drug-Linkers

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Year: 2017
Type: article
Source: Journal of Medicinal Chemistry
DOI: 10.1021/acs.jmedchem.7b00736
Authors: Stephen J. Gregson, Luke A. Masterson, Binqing Wei, Thomas H. Pillow, Susan D. Spencer, Gyoung-Dong Kang, Shang-Fan Yu, Helga Raab, Jeffrey Lau, Guangmin Li, Gail D. Lewis Phillips, Janet Gunzner-Toste, Brian S. Safina, Rachana Ohri, Martine Darwish, Katherine R. Kozak, Josefa dela Cruz-Chuh, Andrew Polson, John A. Flygare, Philip W. Howard
Institutions: Spirogen (United Kingdom), Genentech
Language: English

Topic: Synthesis and pharmacology of benzodiazepine derivatives
Subfield: Organic Chemistry
Field: Chemistry
Domain: Physical Sciences
SDG: Good health and well-being

Open Access status: closed
OpenAlex ID: W2767488985
FWCI: 1.907
Cites: 48
Cited by: 37
Related to: 10
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